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RAD140

Product Information

£39.99

Selective Androgen Receptor Research: RAD140

RAD140 (commonly known as Testolone) is a potent, non-steroidal selective androgen receptor modulator (SARM) engineered for high binding affinity and robust tissue selectivity. Preclinical investigations focus on its unique pharmacokinetic profile, which demonstrates high anabolic activity in skeletal muscle and neural tissues while exhibiting minimal agonistic activity in secondary non-target organs. It serves as an essential analytical reference standard for exploring tissue-specific receptor dynamics and signaling pathways.

Technical & Product Specifications

  • Sample Size: 10 mg / 30 ml (liquid solution)

  • Purity: >98% (HPLC verified)

  • Molecular Weight: 393.85 g/mol

  • CAS No.: 1182367-47-3

  • Solubility: Soluble in DMSO, PEG 400, and ethanol

Pharmacological Mechanisms & Bio-Analytical Applications

Unlike conventional anabolic steroids, RAD140 exhibits a distinct structural profile that prevents conversion into estrogenic metabolites or dihydrotestosterone (DHT) derivatives. Laboratories investigating advanced cellular mechanisms frequently analyze its interactions alongside growth hormone secretagogues. For instance, investigating a rad140 and mk677 stack allows researchers to model synergistic pathways involving both androgen receptor modulation and ghrelin receptor activation in in vitro muscle-wasting and neuroprotection models.

Key areas of academic exploration include:

  • Myotrophic vs. Androgenic Index: Evaluating transcriptional activation ratios in skeletal muscle tissue relative to prostate cells.

  • Neuroprotective Properties: Assessing neuro-signaling preservation, cognitive protection, and androgen-mediated neuronal cell survival in preclinical models.

  • Combination Pharmacology: Measuring the metabolic impact of a combined rad140 and mk677 protocol on cellular turnover, protein synthesis, and nitrogen retention assays.

Sourcing & Laboratory Inventory Standards

When planning compound procurement for institutional laboratories, researchers actively seeking rad140 for sale or looking where to rad140 buy must prioritize third-party mass spectrometry and high-performance liquid chromatography (HPLC) validation. Ensuring verified purity parameters is vital for maintaining reproducibility across complex analytical assays and bioenergetic studies.

High-Purity Reagents by Receptor Chemicals

Receptor Chemicals provides premium-grade research compounds manufactured to meet stringent academic and laboratory standards. Every batch undergoes rigorous quality control protocols to ensure molecular stability and precise concentration consistency for advanced experimental designs.

Description

Selective Androgen Receptor Research: RAD140

RAD140 (commonly known as Testolone) is a potent, non-steroidal selective androgen receptor modulator (SARM) engineered for high binding affinity and robust tissue selectivity. Preclinical investigations focus on its unique pharmacokinetic profile, which demonstrates high anabolic activity in skeletal muscle and neural tissues while exhibiting minimal agonistic activity in secondary non-target organs. It serves as an essential analytical reference standard for exploring tissue-specific receptor dynamics and signaling pathways.

Technical & Product Specifications

  • Sample Size: 10 mg / 30 ml (liquid solution)

  • Purity: >98% (HPLC verified)

  • Molecular Weight: 393.85 g/mol

  • CAS No.: 1182367-47-3

  • Solubility: Soluble in DMSO, PEG 400, and ethanol

Pharmacological Mechanisms & Bio-Analytical Applications

Unlike conventional anabolic steroids, RAD140 exhibits a distinct structural profile that prevents conversion into estrogenic metabolites or dihydrotestosterone (DHT) derivatives. Laboratories investigating advanced cellular mechanisms frequently analyze its interactions alongside growth hormone secretagogues. For instance, investigating a rad140 and mk677 stack allows researchers to model synergistic pathways involving both androgen receptor modulation and ghrelin receptor activation in in vitro muscle-wasting and neuroprotection models.

Key areas of academic exploration include:

  • Myotrophic vs. Androgenic Index: Evaluating transcriptional activation ratios in skeletal muscle tissue relative to prostate cells.

  • Neuroprotective Properties: Assessing neuro-signaling preservation, cognitive protection, and androgen-mediated neuronal cell survival in preclinical models.

  • Combination Pharmacology: Measuring the metabolic impact of a combined rad140 and mk677 protocol on cellular turnover, protein synthesis, and nitrogen retention assays.

Sourcing & Laboratory Inventory Standards

When planning compound procurement for institutional laboratories, researchers actively seeking rad140 for sale or looking where to rad140 buy must prioritize third-party mass spectrometry and high-performance liquid chromatography (HPLC) validation. Ensuring verified purity parameters is vital for maintaining reproducibility across complex analytical assays and bioenergetic studies.

High-Purity Reagents by Receptor Chemicals

Receptor Chemicals provides premium-grade research compounds manufactured to meet stringent academic and laboratory standards. Every batch undergoes rigorous quality control protocols to ensure molecular stability and precise concentration consistency for advanced experimental designs.